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        Pharmaceutical intermediates

        Name

        Key intermediate

        CAS NO
        Axitinib

        3,6-diiodo(1H)indazole

        Methyl 2-mercaptobenzoate

        319472-78-1

        4892-02-8

        Crizotinib

        4-Iodo-1H-pyrazole

        (R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-2-nitropyridine

        4-(4-Bromopyrazol-1-yl)piperidine-1-carboxylic acid tert-butyl ester

        (R)-5-bromo-3-(1-

        3469-69-0

        877397-70-1

        877399-50-3

        877399-00-3

        Lapatinib

        2-(Methylsulfonyl)-ethanamine hydrochloride

        N-[3-Chloro-4-(3-fluorobenzyloxy)phenyl]-6-iodoquinazolin-4-amine

        3-Chloro-4-(3-fluorobenzyloxy)aniline

        104458-24-4

        231278-20-9

        202197-26-0

        Pazopanib

        3-Methyl-6-nitro-1H-Indazole

        2,3-dimethyl-6-nitro-2H-indazole

        2,3-dimethyl-2H-indazol-6-amine

        2,4-Dichloropyrimidine

        3-Amino-6-methylbenzenesulfonam

        6494-19-5

        444731-73-1

        444731-72-0

        3934-20-1

        6973-09-7

        Regorafenib

        3-Fluoro-4-Nitrophenol

        3-Fluoro-4-aminophenol

        394-41-2

        399-95-1

        Afatinib

        trans 4-Dimethylaminocrotonic acid hydrochloride

        848133-35-7

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